Difference between revisions of "Entospletinib (GS-9973)"

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===[[Chronic lymphocytic leukemia]]===
 
===[[Chronic lymphocytic leukemia]]===
# Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. [http://www.bloodjournal.org/content/125/15/2336.long link to original article] [https://pubmed.ncbi.nlm.nih.gov/25696919/ PubMed]
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# '''GS-US-339-0102:''' Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. [https://doi.org/10.1182/blood-2014-08-595934 link to original article] [http://www.ncbi.nlm.nih.gov/pmc/articles/pmc4401348/ link to PMC article] [https://pubmed.ncbi.nlm.nih.gov/25696919/ PubMed] [https://clinicaltrials.gov/study/NCT01799889 NCT01799889]
  
 
==Also known as==
 
==Also known as==

Revision as of 18:21, 27 June 2024

Mechanism of action

Spleen tyrosine kinase (SYK) inhibitor

Preliminary data

Chronic lymphocytic leukemia

  1. GS-US-339-0102: Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. link to original article link to PMC article PubMed NCT01799889

Also known as

  • Code name: GS-9973