Difference between revisions of "Entospletinib (GS-9973)"

From HemOnc.org - A Hematology Oncology Wiki
Jump to navigation Jump to search
(Created page with "=Mechanism of action= Spleen tyrosine kinase (SYK) inhibitor =Preliminary data= ==CLL== # Sharman...")
 
m (Text replacement - "http://www.ncbi.nlm" to "https://www.ncbi.nlm")
Line 5: Line 5:
  
 
==[[Chronic_lymphocytic_leukemia_(CLL)_and_Small_lymphocytic_lymphoma_(SLL)|CLL]]==
 
==[[Chronic_lymphocytic_leukemia_(CLL)_and_Small_lymphocytic_lymphoma_(SLL)|CLL]]==
# Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. [http://www.bloodjournal.org/content/125/15/2336.long link to original article] [http://www.ncbi.nlm.nih.gov/pubmed/25696919 PubMed]
+
# Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. [http://www.bloodjournal.org/content/125/15/2336.long link to original article] [https://www.ncbi.nlm.nih.gov/pubmed/25696919 PubMed]
  
 
[[Category:Drug index]]
 
[[Category:Drug index]]

Revision as of 03:07, 2 December 2016

Mechanism of action

Spleen tyrosine kinase (SYK) inhibitor

Preliminary data

CLL

  1. Sharman J, Hawkins M, Kolibaba K, Boxer M, Klein L, Wu M, Hu J, Abella S, Yasenchak C. An open-label phase 2 trial of entospletinib (GS-9973), a selective spleen tyrosine kinase inhibitor, in chronic lymphocytic leukemia. Blood. 2015 Apr 9;125(15):2336-43. Epub 2015 Feb 18. link to original article PubMed